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ÀÛ¼ºÀÚ ´ÚÅÍÄÚ¸®¾Æ Á¶È¸¼ö 3804
¥°, Metronidazole, Mupirocin, Polymyxin



1. Metronidazole

nitroimidazole°è Ç׿øÃæ ¾àÀ¸·Î Çø±â¼º ±×¶÷ À½¼º°£±Õ(G(-)°£±Õ), Çø±â¼º G(+)±¸±Õ,°£±Õ, ¹× Æ®¸®Äڸ𳪽º¿¡ ´ëÇØ ±¤¹üÀ§ È°¼ºÀ» º¸ÀÌ´Â ¾à¹°ÀÌ´Ù.

°æ±¸, IV, ÁÂ¾à µîÀÇ ÇüÅ·ΠÅõ¿©µÇ¸ç BBB¸¦ Àß Åë°úÇÏ°í ħ, ´ãÁó, ´¢, À¯Áóµî¿¡¼­µµ ½Å¼ÓÇÏ°Ô À¯È¿ ³óµµ¿¡ µµ´ÞÇÑ´Ù.

¼ö¼úÈÄ Çø±â¼º±Õ °¨¿°ÁõÀÇ Ä¡·á ¹× ¿¹¹æ¿¡ »ç¿ëÇϸç trichomonas³ª bacterial vaginosis, ³úÁ¾¾ç Ä¡·á¿¡ ÀÀ¿ëµÈ´Ù. ±¹¼Ò¿ëÀ¸·Î Gel typeÀÇ Á¦Á¦µµ ÀÖ´Ù.

warfarinµîÀÇ Ç×ÀÀ°íÁ¦ÀÇ ÀÛ¿ëÀ» Áõ°¡½ÃÅ°°í disulfiram°ú °°Àº ÀÛ¿ë ¶§¹®¿¡ alcohol°ú ÀÇ º´¿ëÀ» ±ÝÇÑ´Ù. »ç¶÷¿¡°Ô¼­ ŹÝÀå¾Ö¸¦ ÃÊ·¡ÇϹǷΠÀӺο¡°ÔÀÇ Åõ¿©¸¦ ±ÝÇÑ´Ù.



2. Mupirocin

Pseudomonas fluoresens¿¡¼­ »ý¼ºµÇ´Â natural productÀÌ¸ç ±¹¼Ò¿ë ¿¬°íÁ¦·Î¸¸ »ç¿ëÇÏ´Â ¾à¹°ÀÌ´Ù.

mupirocinÀº Isolecyl tRNA synthesis¿¡ °¡¿ªÀûÀ¸·Î °áÇÕ, ±ÕÀÇ protein synthesis¸¦ ¾ïÁ¦ÇÏ¸ç »ç¶÷ÀÇ Á¤»ó¼¼±ÕÃÑ¿¡´Â ÀÛ¿ëÇÏÁö ¾Ê°í G(+)±¸±Õ¿¡ Àû¿ëÇϸç Staphylococcus, Streptococcus, E.coli, Hemophilus influenzaµîÀÇ ÇǺΰ¨¿°¿øÀαտ¡ »ç¿ëÇÑ´Ù.



3. Polymyxin B

PolymyxinÀº G(-)±Õ¿¡ ÀÛ¿ëÇÏ´Â ¿°±â¼º peptidefb·Î ½ÅÀ嵶¼ºÀÌ °­ÇØ polymyxin B, E ¸¸ÀÌ »ç¿ëµÇ°í ÀÖ´Ù.

polymyxin B´Â º¸Åë polymyxin B sulfate formÀ¸·Î ¼ö¿ë¼º, ¾ÈÀü¼ºÀ» ³ô¿© »ç¿ëÇÏ¸ç ¼¼Æ÷º® ±â´ÉÀ» ¼Õ»ó½ÃÄÑ ¼¼Æ÷³»¿ë¹°À» ¿ëÃâ½ÃŲ´Ù. Pseudomonas¿¡ ³ôÀº È°¼ºÀ» º¸ÀÌ°í endotoxinÀÚüµµ ºÒÈ°¼ºÈ­ ½ÃŲ´Ù. G(+) ¹× Proteus, Neisseria ±ÕÁÖ¿¡´Â °¨¼ö¼ºÀÌ ¶³¾îÁö°í ³»¼ºÀº Àß »ý±âÁö ¾Ê´Â´Ù.

½Å°æµ¶¼ºÀ̳ª ½ÅÀ嵶¼ºÀÌ °­ÇØ Àü½ÅÀû¿ëÀº ÇÏÁö ¾Ê°í ±¹¼ÒÀûÀ¸·Î Á¡¾È¾×À̳ª ¿¬°í·Î »ç¿ëÇÑ´Ù.



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